Carperidine

Carperidine
Identifiers
	IUPAC name ethyl 1-(3-amino-3-oxopropyl)-4-phenylpiperidine-4-carboxylate;
CAS Number	7528-13-4 ;
PubChem CID	24149;
ChemSpider	22571;
UNII	LZ6E4G9827;
ChEMBL	ChEMBL2104584;
CompTox Dashboard (EPA)	DTXSID10226254 ;
Chemical and physical data
Formula	C17H24N2O3
Molar mass	304.390 g·mol−1
3D model (JSmol)	Interactive image;
	SMILES CCOC(=O)C1(CCN(CC1)CCC(=O)N)C2=CC=CC=C2;
	InChI InChI=1S/C17H24N2O3/c1-2-22-16(21)17(14-6-4-3-5-7-14)9-12-19(13-10-17)11-8-15(18)20/h3-7H,2,8-13H2,1H3,(H2,18,20); Key:IXZCNCWEDOHVLK-UHFFFAOYSA-N;

Carperidine (Carbamethidine) is an opioid analgesic drug related to meperidine. It has analgesic and antitussive effects with similar potency to codeine, though several related compounds are significantly more potent.^[1]^[2]^[3]

References

^ US 117139, Aram M, "4-aryl-1-carbamylalkyl-piperidines.", issued 7 January 1964, assigned to Sterling Drug, Inc..
^ List PH, Hürhammer L (1973). "C, Sachverzeichnis für die Bände I–III, VIIA". Hagers Handbuch der Pharmazeutischen Praxis (Für Apotheker, Arzneimittelhersteller Ärzte und Medizinalbeamte). Vol. 1, 2, 3, 7A. Berlin, Heidelberg: Springer. pp. 56–82. doi:10.1007/978-3-642-67660-4_3.
^ Richards GC, Sitkowski K, Heneghan C, Aronson JK (October 2021). "The Oxford Catalogue of Opioids: A systematic synthesis of opioid drug names and their pharmacology". British Journal of Clinical Pharmacology. 87 (10): 3790–3812. doi:10.1111/bcp.14786. PMC 8518704. PMID 33608948.

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[1] US 117139, Aram M, "4-aryl-1-carbamylalkyl-piperidines.", issued 7 January 1964, assigned to Sterling Drug, Inc..

[2] List PH, Hürhammer L (1973). "C, Sachverzeichnis für die Bände I–III, VIIA". Hagers Handbuch der Pharmazeutischen Praxis (Für Apotheker, Arzneimittelhersteller Ärzte und Medizinalbeamte). Vol. 1, 2, 3, 7A. Berlin, Heidelberg: Springer. pp. 56–82. doi:10.1007/978-3-642-67660-4_3.

[pmid33608948-3] Richards GC, Sitkowski K, Heneghan C, Aronson JK (October 2021). "The Oxford Catalogue of Opioids: A systematic synthesis of opioid drug names and their pharmacology". British Journal of Clinical Pharmacology. 87 (10): 3790–3812. doi:10.1111/bcp.14786. PMC 8518704. PMID 33608948.

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Identifiers

IUPAC name ethyl 1-(3-amino-3-oxopropyl)-4-phenylpiperidine-4-carboxylate
CAS Number	7528-13-4^Y
PubChem CID	24149
ChemSpider	22571
UNII	LZ6E4G9827
ChEMBL	ChEMBL2104584
CompTox Dashboard (EPA)	DTXSID10226254
Chemical and physical data
Formula	C₁₇H₂₄N₂O₃
Molar mass	304.390 g·mol⁻¹
3D model (JSmol)	Interactive image
SMILES CCOC(=O)C1(CCN(CC1)CCC(=O)N)C2=CC=CC=C2
InChI InChI=1S/C17H24N2O3/c1-2-22-16(21)17(14-6-4-3-5-7-14)9-12-19(13-10-17)11-8-15(18)20/h3-7H,2,8-13H2,1H3,(H2,18,20) Key:IXZCNCWEDOHVLK-UHFFFAOYSA-N

Carperidine

See also

References